



| 货号 | 包装规格 | 操作 |
|---|---|---|
| SML0921-5MG | 5 mg | |
| SML0921-25MG | 25 mg |
≥98%(HPLC)
AR7 has been used:
as chaperone-mediated autophagy (CMA) activator to study the activity of CMA in rat liver lysosomesPMID 30610733as a CMA activator to study its effects on expression of DEAD-box helicase 3 X-linked (DDX3X), eukaryotic translation initiation factor 4A1 (EIF4A1), and eukaryotic translation initiation factor 4H (EIF4H) in cancer cellsPMID 30821613to study its effects on synuclein α (SNCA) oligomer levels in mature primary cortical neuronsPMID 30983487
AR 7是一种非典型的视黄酸受体(retinoic acid receptor,RAR)α拮抗剂。
AR 7是一种非典型的视黄酸受体α(retinoic acid receptor α,RARα)拮抗剂,近年来发现,通过RARα的信号传导抑制了分子伴侣介导的自噬(chaperone mediated autophagy,CMA),阻断RARα的信号传导对CMA有促进作用,但能抑制巨噬细胞的自噬,AR 7只拮抗CMA的抑制作用,而不影响巨噬细胞的自噬,使RARα对自噬的两种作用得以独立研究。
| 英文名称 | AR7 |
| CAS 号 | 80306-38-3 |
| 经验分子式 | C15H12ClNO |
| 分子量 | 257.71 |
| UNSPSC | 12352200 |
| NACRES | NA.77 |
| InChI key | 普什图市KBDGXBB-UHFFFAOYSA-N |
| SMILES字符串 | 碳酸氢钠 |
| 含量测定 | ≥98%(HPLC) |
| 形态 | 粉末 |
| 颜色 | 白色至米色 |
| 溶解性 | DMSO:20 mg/mL,澄清 |
| 储存温度 | 2-8°C |
| 质量等级 | 100 |
| 包装规格(货号 SML0921-5MG) | 5 mg |
| 包装规格(货号 SML0921-25MG) | 25 mg |